Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3412	CP-135807 CAS No.151272-90-1	CP-135807/CAS No.151272-90-1 is an orally active and selective 5-HT1D agonist (IC50=3.1 nM), bovine). CP-135807 mediates central psychoactivity and can be used in antidepressant research.	price>
R-R-3413	Vortioxetine-d8 CAS No.2140316-62-5	Vortioxetine-d8/CAS No.2140316-62-5 is a deuterium labeled Vortioxetine. Vortioxetine is an inhibitor of 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT, with Ki values of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively.	price>
R-R-3414	Isopteropodine CAS No.5171-37-9	Isopteropodine/CAS No.5171-37-9 is heteroyohimbine-type oxindole alkaloid components of Uncaria tomentosa (Willd.) DC. Isopteropodine acts as positive modulators of muscarinic M1 and 5-HT2 receptors.	price>
R-R-3415	Anpirtoline hydrochloride CAS No.99201-87-3	Anpirtoline hydrochloride/CAS No.99201-87-3 is a hydrochloride of anpirtoline. Anpirtoline is a agonist of 5-HT1B.	price>
R-R-3416	Lurasidone-d8 CAS No.1132654-54-6	Lurasidone-d8/CAS No.1132654-54-6 is deuterium labeled Lurasidone. Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7 with IC50s of 1.68 and 0.495 nM, respectively. Lurasidone (SM-13496) is also a partial agonist of 5-HT1A receptor with an IC50 of 6.75 nM.	price>
R-R-3417	Loxapine-d8 CAS No.1189455-63-7	Loxapine-d8/CAS No.1189455-63-7 is the deuterium labeled Loxapine.	price>
R-R-3418	(S)-Renzapride	(S)-Renzapride ((S)-BRL 24924) is the isomer of HY-14147 Renzapride. Renzapride is a 5-HT4 receptor agonist with a Ki value of 115 nM. Renzapride also is a 5HT2b and 5HT3 receptor antagonist. Renzapride can be used for constipation predominant irritable bowel syndrome (C-IBS) study.	price>
R-R-3419	Cyclobenzaprine-d3 hydrochloride CAS No.1184983-42-3	Cyclobenzaprine-d3 (hydrochloride)/CAS No.1184983-42-3 is the deuterium labeled Cyclobenzaprine hydrochloride. Cyclobenzaprine hydrochloride (MK130 hydrochloride) is a skeletal muscle relaxant and a central nervous system (CNS) depressant.	price>
R-R-3420	LY 344864 S-enantiomer CAS No.186544-27-4	LY 344864 S-enantiomer/CAS No.186544-27-4 is the S-enantiomer of LY344864. LY344864 is a 5-HT1F receptor agonist.	price>
R-R-3421	Perphenazine-d4 CAS No.155593-75-2	Perphenazine-d4/CAS No.155593-75-2 is the deuterium labeled Perphenazine. Perphenazine is a typical antipsychotic agent, inhibits 5-HT2Areceptor, Alpha-1A adrenergic receptor, Dopamine receptor D2/D3, D2L receptor, and Histamine H1 receptor, with Ki values of 5.6, 10, 0.765/0.13, 3.4, and 8 nM, respectively.	price>

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